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氯氮平的严重不良反应

2017-10-24 8页 doc 31KB 15阅读

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氯氮平的严重不良反应氯氮平的严重不良反应 2006??2?)?L3???L05?%?????d???? ?M?A?????u???H?????? ?d????(???i?2?????????m?t??272600) ?M?A???M???????A???????C???????????-???B???m???/?? ?????P?????????-???F?P?????TD1,D2???????)?-?????D?? ??5-HT2?????????BE0?????T???P???P?????????????????? ???)E0...
氯氮平的严重不良反应
氯氮平的严重不良反应 2006??2?)?L3???L05?%?????d???? ?M?A?????u???H?????? ?d????(???i?2?????????m?t??272600) ?M?A???M???????A???????C???????????-???B???m???/?? ?????P?????????-???F?P?????TD1,D2???????)?-?????D?? ??5-HT2?????????BE0?????T???P???P?????????????????? ???)E0?????F???5????E2????E2???w?0?sE2???%???????????D ????????E0?????D???????????????????B?????m???u???’???? ?????????w?????????????1?????G?????-?????B?????D?X???? ????????E0???M?A?????4???????????m?-?????????????u???? ???????D????E0???(?????????A???????u???H?????????????,?- ???4???t????????????E0 1???m?? ?????????????????5?w???G?-35???-?????-???[?????- ?t??????????:?m?hE2???????mE2????????????E0?????? ???w?????(????E0?????????????-????????????E0?????? ?s?-????X???:???????Y??E2?m?Y??E2?D?G?s???????????0 ?sE0?????T?D?B?M?A??25mg?-2?[.d??hK?-?T?X?????????- 2???T??????400mg.d-’?-???2?B??E0?????%?????2?????? ????1??2?[?-?????????B???s?6????E0?B?B???L42?l???- ???5???F????????????E2????E2????????E2?g?E?-?????? ?m???:?????2?-???????w8/4KPa?-????140?[/minE0???% ?D???????G?m??????????;????E2???GE2????E2?????-?B 5%?????9?????3???-5%??10%???3???-???(??????????E2 ?P???????3????E0??????1h?T?????1???E13/6KPa?-???? 102?[/min?-?????D???-???5?????????-?D???%E2?I???? ???-????????600m1?-???????????2?????????-??2h?T?? ?5?????????,???-???w6/4KPa?-???s?u???d?????-???7?x ??E0???????G?G?????-???????????????-?????B???s???? ??E2?w?????????????-????????E0?????????g????????6h, ?????????M?A?????H???(?G???????G?m???-????E0 ???D??[21?????????G?-23???-1997??5?)26???????????- ?????w:?(???O???????-?????????????????????0?s?-?n?? ?M?K?????)?Y?m???????-20?l?T???????H?(???-?o?B?M?A?? ?????-?????????w25mg?-3?[.d-hK?-20?l?T????125mg, 3?[.d-,?-????50?l?T???????????U???-8?)7?????F?????? ??E2????E0????:?????5?-???l??39.5[6?-???????-?? ???????-??????????II?????G?-?????D?.?G?(?????-???:?? ?,205cm?-?????,4??5cm?-?D?????-?????-?u????:?? ????3600/mm3?-?<?G67%?-????33%?-??????:II:25u, ??????????:???m?????-SGPT:145u,B?????????w: ????????6.6cm?-????5.lcm?-????????16.lcm?-????8. 6cm?-?????H???-?????-???:???GE0?????????-???????% ???-????E2???????6???M?2?????-?????H???????-?????6 ?X?X?,???-?E8?)15???-??????????1000/mm3?-?????H ???-???.???P???6???w?u?????<???G?????-???????????-?? ?????????w?????????w:c??????D?s???????%?t??E0c??????? ????????????E0c??????????????%?t???-???<E2??E2?? ?????????%?w?t?-???D???P???s?(??E0c????????????????? ???P?-???D?(???H?T?????-???????B???-???????????-?? ?????-?G???(?????E?s???-?P???????-???????X?X?????-?? ???2???????????????R?-??8?)18??????E0 ???o??[31????12?????5???[?H?M?A???-???????B50mg/ d?-???H???T3??5?:?????%?:??E2?m??E0???<?O4??E2??8 ???-50?????14??E0?m???5?????w?:???G?C?-???s?u???-?? ???????-???h???????-???Y???w???G???????%E0?:???5???? ?w???F???g?-?????????-?????????-???2???h?-???Y???? ?w???G???????.E0????????E2?????????-1??3?:???T???H ???sE0 ???-??[a1????3?????5???H?:?????M?A???T(G50mg/ d)???%?m??E0?????????????d???-?M?A?????????????B?? ?G?>?????0?-???P??????10?H???1E0???M?C???G?xE2????E2 ????E2?m?????0???????-?????t?????9?????????hP450?t?G ?B?>???????B???G???x?-?-???G?????C???5?????t?G?????? ???-???.???%?m??E0???’?-?M?A?????D?????,???t??5-HT, ???1???h???????B?-?.?4???????G??????E0???Y?????w(?H ?B?M?A???T)?-???5?????????????E???F?-?.???%?m??E0 2?u???’?????? ??????[51????28.7%?????5???%???u???’??????E0?t???? ???w?????7??E2???????.?-?????????-????E2????E2???h ??????E0???T?M?A???t?????B?????????P???P?????????D??E0 ?????????????????H??????[61?t???M?4??????????????E2 ?????????????????????????m???H??????E0?????????????7 ??:???????t??>10x109/L;?????????????7??:???? ???t??<4x109/L?-???????????m?7??:????????/???? ????<75%E0?????’?????????-100?????5?H?B?M?A?????? 4???-??????????1?[E0???<?-?O58???-??42???-?????? ??33.7??18.3??E0???????w125--500mg?-????270.0??187. 5mgE0????:?????????P14??(14%)?-?????????m20?? (20%)?-?????????m2??(2%)E0???D?????-???????w ?????%??0.16%?-?C???m???????????????P???%???w25%, ?????????m???%???w9.34%E0?t?????w?T???5???0???????? ?B?-?B???T???%???2?????D???-???’?B?????????G(> 400mg/d)???M???%?H????????????????E0 3?????? ?,????[c,1?????-???G???51???-39???-?B?B??(400mg/ d)17?l?T?-?????s???????-ALT??AST?(?x????5817.83 u/L??2550.51u/L?-???B?M?A???-???????????????-?X?X ???H???sE0???w?M?A???????9?????????hP450?t?G?B???5?? ???????????-?h?X???????<?M?A?????????9?????N?M?A?????? (?,??41) MEDICINEINDUSTRYINFORMATION.?P???????? 2006??2?)?L3???L05?%?R???d???? 34?????m???c?)???,?/?m???c?R???(?? ??????(?????2?s?????t??364100) ?m????10???????F???,?/?m???c???534???-?B???????, ?<???????????????-???t?????,: 1?R?????? 1.1???L?????O28???-??6???-????19--77???-?? ??37.5??E0 1.2?????T?????DGCS?(???-3-8?(20???-9--12 ?(9???-13??15?(5??E0?:?????????????w???h?????1??E2 ????E2?P???:???H??E025???????w?<???G?????-???l?2?? 40[6???1?-3???w???l?H??E034?????????D?H?-?,?????R?? ???9?????-?????w???l???-?R???????R?<???’?<???G?????? ???)???-?u?G?1???’??????24???-?????9?1??21???-???< 2?????????8?G?????????????:??E0 1.3??????????34???????????R??CT?????-?????? ??????10???-?m?x?c19???-????E2?m?????c3???-?u?x?G ?m????1???-?????’?c?G???????,??????1??E0 1.4???????????????5???M9???-???????????????? ?M6???-???????????????????-??19???u?????m???c?R?D?? ???-???:?????,?/?m?????5?????????l????E0?1???’?????? 24???-???%?????????-?s???????????????-?s?????D???3 ???????-????????????????????????E0???l?????5???H?B?? ?9??????;???l???u???5???B???????l?????3?????????3E0 ???)?????????K?B?????C?R???????????-???-???????????? ???-???8?G?????????????:???P???B?????????G?m???-???? ?1?????%?????m????????????E0 1.5?????o??Glasgowoutcomescale?7???-????6 ???-?H???%??1???-????3???-?<??9???-????15??E0 2???? ?/?m?,?????c?w?????G???????G?c???-???5?m???-?? ?/?m?,?????????E?a?c?-?T?5?K?s?M?B?u???????m???c?? ???1?????????????-?m?R???-???????????-?m???????? ???m?????T?-?????/?m?,?????????E?????-???-???%?? ???G?w???G????E0 ?????,?/?m???c?t???R???????w?:???????P???:???-?? ?l?6??????(???????w?t)?-?R?????9????(?????l???? ?w????)?-?1???’???????-???8?G?????G?????????:??E0 ?P???/?m?,?????c?????C?????????-???c?w?F?H???-???? ?)???m???????????c?-?/?m?,???c?????s??????E0?????- ?????D???c???????G???????-?C?????E?/?m?,?????c???? ???-???M???u?????m???c?????-?s???????????????1???- ?C???G?P?????5?)???D?????????m???c?-???????????????) ?????????KE0?N?????????????m?R???????????????????M?? ???????A?-?-?????M?N???/?m?,???????G???c?????A????E0 ?/?m?,?????c?????????????-?R?????9?????-???’???????- ???8?G?????????????:???M???????????T?????????h?-???? ??????E0?????R?D?????5?-?6???w?,?/?m?????????l?<?? ?????????-?????l?????c?????w?????????-?????????m?8 ?G?????????(???-???????<???-???2???s?m???????????? ???9?-???????????m???????R??E0?%?(?????,?-?,?/?m?? ?F?????????(??ACTH???????T???(??ADH?-?P???????? ???’???<?Y???B???8?:?????6???-???-???2?w?????s?R???? ?9E0???s???2?,ACTH??ADH???2???2?????-???,?/?m ???c?c???M???1?s???????s???E?????????????C?6?-???-?? ?????l???-?R???????R?<???’?????????)???-?R???1???o ?????????????2?R?Y???B?????????2???????U??E0 ?u?????m???c?????s???????’???????-?D???????????% ??????90%?-???’???????????w?(?????P???????????-???H?? ?????1?????????E???t?????B?-?R???1?????????’?????????? ???-???E???????-??????E0???8?G?????????????:???M?????8 ?:???-?????????????R?G?w?????-???%?w?(?T?,?/?m???????? ?????’???????c?D???-?????????????-???8?:???-?????B???? ?h?????-?????????????????h???%?-???????:???w??E0?? ?I???’???/?? (?1??62??) ????E0?????B?????,?<???7???:???s?????’?-???u?e?? ?F?????B??E0 ???6???A !??????.?B?a?A????????????????1??.?<???t???????????- 2001?-21(7):448. 2???D??.?B?a?A?????????????w?????)???<???G?????w?(?? ???<???????-2002,16(9):574. 3???o???-??????.?????:?????a?A?????m??12???(??.?<?? ???)?-2000,3(1):25. 4???-??.?:?????a?A???4???m???????B3??????.?1???????t ???-1998?-6(2):84. 5???????-?/????.?a?A???H????????????.?<???????????- 1997?-32(9):561. 6??????.?a?A?????u???H??????.?<???????-2003,17 (4):260. 7?,?????-?????N.?a?A???????????0?s.?????H???????????- 1999?-1(2):117.?? ?I???’?????5?? MEDICINEINDUSTRYINFORMATION?t?????P????41
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