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复方柳氮磺吡啶栓的制备及临床应用

2017-09-02 8页 doc 27KB 25阅读

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复方柳氮磺吡啶栓的制备及临床应用复方柳氮磺吡啶栓的制备及临床应用 2006??12?4?R3???R35?X???????g???? ?8?????>???????Q???]?(???<?????y ?B?s???%?????N?%?B?? (?????2?????e?????R???????e???%????????453100) d;????dI????:?]???8?????>?????>?Q???]?(???????y?????]?????%???????<??????d0??? ?:???y?5???????...
复方柳氮磺吡啶栓的制备及临床应用
复方柳氮磺吡啶栓的制备及临床应用 2006??12?4?R3???R35?X???????g???? ?8?????>???????Q???]?(???<?????y ?B?s???%?????N?%?B?? (?????2?????e?????R???????e???%????????453100) d;????dI????:?]???8?????>?????>?Q???]?(???????y?????]?????%???????<??????d0??? ?:???y?5???????????? ???>?????>???=???%????110???????H?????????3?????<??????????d0????:???>??? ??>?=???????%?y???????%?? ?????H???????????4???r65.0%?%?e?)?????r86.7%d0????:?1???????4?5?%?y???????????%?&l t;?????????(d0 d;???>??I?8?????>?????>??;?]?(;?y?????];?<?????y ???>?????>?r?????????????%?e???y???????????H?? ????(UC)?%???G???5?r???G???Q?G?/??d0?8?????>?????>?Q ?????>????Q?r?e???%?????J?????????????]?;???Q?%?? 110???????H?????????3?????<???????????%???7???>???? ?????????????%?????8?????>????0?Q???????(?%???y?? ???%?w??????d0 ?%?1?????]?( 1.1?1?? ???>?????>50g,?J????????????1g,????????4000 119.8g,????????600012g,?-?9??5.4g?%?i??11.8g?%???] ?;100??d0 1.2?]?( ??????????4000??????????6000?%???<???:?????? ?9?%???S??????5092?%?????i?????-?9??d2?J????????????d2 ???>??????????(?????m????????)?%???X?3?????????5???% ?????Q?M?P?%?????%?>???%?????3??????d0 2?y?????] 2.1?H?? ?R???r?;???????h???Q?G?%?????%????d0 2.2??Nil ???R???0??(???????????>?????>120mg)?%?(???%???? ????10ml,?3???%?????%??????2ml?%???%????0.2g?%?Q?Q?? ???%?v?c?;?????????Ed0 ???=?????????.???????%???=?9???????5????????(d:?P ??????d.2005????????????WA)?????%?y359nm?????1?) ???H?s?]d0 2.3???? 2.3.1???????0?p?4?Q?G???.(d:?P??????d.2005?????? ??????ID)???????0??????????d0 2.3.2????????????????????????(d:?P??????d.2005?? ??????????XB)?????%?p?4????d0 2.3.3???X???????????X????????????(d:?P??????d. 2005????????????MJ)?????%?p?4????d0 2.4?=?????? 2.4.1???????????R??10???%?????????%?(???%?????%???? ?????0??(???????????>??????0.15g)?%??200ml?????P?% ??0.1mol/L?J?H?9??????20ml?%?????<???P?%?-?????????% ?c???????S?%???<???e???%?????%?????%??????????????2 ml?%??200ml?????P?%???????????????Q????(pH4.5)20ml, ?y?<???????e???%???<???????%???=?9???????5???????? (d:?P??????d.2005????????????WA)?%?y359nm?????1?? ???s?]???%?)C18Hi4N40yS???s?]?????r658????????d0 2.4.2???????????=?????????.?????%?5?=?????R??3???a ?????=??(??1)o ??1?)???a?????=f????????(n=3) ?a?????????>?????> ?(?r??(%)RSD(%) 050326 050420 050518 99.8 99.9 99.8 0.45 0.30 0.66 2.5?x???H???? ?53???a???y?s?S?.?????????%?c??1???%???9??d2?? ??d2???????????????9?%?e???=???????7?c???9?%???7?R?? ?x???H????d0 3?<?????y 3.1???R???? ?<??UC???3110???%?a66???%??44??d0???????I16 ???%???H68??d0110?????3?P?)?????????5?h???9?<?????? ???????r???5?=?r:???????????v?<???378???%??71%;?? ???357???%??52%;?????3103???%??94%;????64???%?? 58%;????24???%??22%;???L?7??46???%??42%;???????? 98???%??89%d0?v?)?????????????????H??????d2???G???? ????d2???????????????7???????%?g??????????????????d0 3.2?<???????5?? ??????60???%??????50???%?/???v???????????y?H ?=d2???????<???????????????R???%?%??:?????%?/?????0?? ?c?????0(P>0.05)?%???)?????Hd0 3.3???????? ???????9?y?8???>?????>?Q?%???M1??,1-2?M//d;?? CHINAMEDICALHERALD?????e???b??157 2006??12?4?R3???R35?X ???????8???>?????>??(?:?????:?)?????m?)??????)?%?? ?M1.5g,3?M/d,6??1???.d0 3.4?????/???(?? ???4:?<?????????E?%?H???s?????????s?%?????????= ?????????8???sd0 ?)??:?<?????????R???E?%?H???s?????????s?9?????0 ?s?%?????9???G???????????.??????d0 ????:?<??????d2?H???s?????????9???G???????f????d0 3.5???????? ??????60???%??????50???%????2?f???.?????%?h???? ???/???(???%???????????7?c?i????????(??2). ??2???????7?????????????? ???=???? ?e???????4?)?????? ?e?)???? % ?%J ld2 ~ 1 1 2 9 2 ?? J ??. 1 60 50 ?????? ?????? 96.7 74.0 x2=5.66,P<0.05 4???? ?????H?????????????r?]?m?8?b?5?3???%?????7????Pl ???Bd2?X??d2???????????????e???)??CAd0???????????5?? (CD44?ad2???H?9?>(N???7UC???X???????????d????????d0 ?J???????????????????v??(?/???-???v??)???Wd2?h ????????d2????d2?Q??????d2????????d0 ?1???P?????y?????-?9?????r?s???%?x???H????d0 ???????????X?5???y?%?????S?8???9?????Q?Q?????? ???P?%?????c?<???H?????%???????c?????H????d0?y?????? ?????y?]?;???Q?G?????????7???s?]???y???y???4?;?0?? ???0???y?]????d0 ???>???????????Q?G?7???8???G?????%???)?????8?? ????pH?9???<??d2???????8???????I???????y?<??d2???U ?????????I?????????yd2?s?]?????Ud2???y??????d2??????d2 ??????????????d0 [???6???>] [1]???????%?????7?%?c?????%??.?????8?4?????????H???????????????y [a]???????9?G???%1998,6(1):87. [2]?E?????%?????g.???????????)?????????????H??????[[J].???????9?G ???%1998,6(8):705. [31CollinsCE,CahiilmrNewlandAC,etal.Plateletscirculateinanactive stateininflammatoryboweldisease?d.Gastroentorology,1994,104(4):840. [4]???)?%?,?4???%?????m?????X?????H???????b?????????H?9?>???? ?X?????I???d?P?????9?????G???%1998,15(5):289. (?]?u???X:2006-10-08) (?:???R162??) ?-???????????????????B????d0 ?R???????c?r:AMI,UAP??DD,Fg?=???7?c???????? ????????SAP???%?gAMI???=??????UAP???%?-?E?????? ???)?e???????<??d2???vd2???;???I?v?Q?%?%???????H???? ???????e?%???????????????m?v??d0Fg?????7???????????; ?)??d0UAP??AMI???%???????v?-???????)?v?Q???;?%???v ?Q?8?????????e?????????rUAP?%?%???]?????e???????? ?rAMI.UAP???3???????%???????????v???2???8?d???]?% ?l?????rAMI.AMI???3???)???)???r?????????????y?%?v ?Q???;???X???????%????DD?=??????d0?????%DD?=???????% ???r?????????XAMI???????H???H?%?7?)?????>????????d0 UAP??DD?<?H?3??Fg?<???7?c?U???x?H?3?%?%AMI,SAP ???/????Fg?<???????c?????0?%???7?????5UAP???3???? ?-???v?Q?r?e?????5???B?%?????????)???W?9?0?y?????? ??d2???H?????Bd0??UAP???3Fg?<???????%?%DD?<?H???? ?I?-?p?)?????????????B???y?%?????0?v??d2???u??d2???v ??d2?s????d0 ?R????????????:SAP???PDD,Fg?=???%?????????? ???8?????%???????????I???%???7?1???????,???????)?? ?Wd2?????H?N???????-?e???????%???)?H???v?Q???;?%???? ?????e?H???h???%?%?8?G??????DD,Fg?=???7?c???????? ???????s???%???7DD?w?????%?v???????.???????%?6???? ???%??????????d0?????%DD?=?????????)???????=?8?G???? ?????y?%?????<?????X?????8?x?????????????????????? ?????????)?????I??d0 ?R???????c?r?%DD???r????????d2????d2???Xd2?????? ???B???v?e?H???????e?H???(?(?%???4Fg?<???5???%???? ?8?G?????????=d2?/????????????d2?(???????????7?????? ?)???????<?????wd0 (?]?u???X:2006-11-12) 158??.????????CHINAMEDICALHERALD
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